Publications

2017

« Synthesis of 1,4-disubstituted 1,2,3-triazole Derivatives Using Click Chemistry and their Src Kinase Activities »
A. LEBEAU, C. ABRIOUX, D. BENIMELIS, Z. BENFODDA, P. MEFFRE
Medicinal Chemistry (2017) 13 (1), 40-48. DOI: 10.2174/1573406412666160404125718
IF(2015)=1,363

2016

« Advances in the synthesis of α‑quaternary α‑ethynyl α‑amino
acids »
T. BOIBESSOT, D. BENIMELIS, P. MEFFRE, Z. BENFODDA
Amino Acids (2016) 48:2081-2101 (published online 16 june 2016). DOI : 10.1007/s00726-016-2276-2
IF(2015)=3,196

« Spatial distribution of triazine residues in a shallow alluvial
aquifer linked to groundwater residence time »
L. SASSINE, C. LE GAL LA SALLE, M. KHASKA, P. VERDOUX,
P. MEFFRE, Z. BENFODDA, B. ROIG
Environ Sci Pollut Res (2016), in press (published on line 22 july 2016). DOI : 10.1007/s11356-016-7224-x
IF(2015)=2,760

« Synthesis of a Novel Rhizobitoxine-Like Triazole-Containing Amino Acid »
T. BOIBESSOT , D. BENIMELIS, M. JEAN, Z. BENFODDA, P. MEFFRE
Synlett (2016) 27 (19), 2685-2688. DOI: 10.1055/s-0036-1588300
IF (2015)=2,323

« The rational design, synthesis and antimicrobial properties of thiophene derivatives that inhibit bacterial histidine kinases. »
T. BOIBESSOT, C. ZSCHIEDRICH,  A. LEBEAU, D. BENIMELIS, DUNYACH-REMY, C. , J.-P.  LAVIGNE, H. SZURMANT, Z. BENFODDA, P. MEFFRE
J. Med. Chem. (2016) 59 (19), 8830-8847. DOI: 10.1021/acs.jmedchem.6b00580
IF (2015)=5,589

2015

« Ethynylglycine synthon, a useful precursor for the synthesis of biologically
active compounds : an update. Part I : preparations of ethynylglycine synthon »
Z. BENFODDA, D. BENIMELIS, G. REGINATO, P. MEFFRE Amino Acids (2015) 47:271–279 (published online 07 january 2015). DOI : 10.1007/s00726-014-1902-0. IF(2014)=3,293

« Synthesis, resolution, and determination of absolute configuration
of protected α‑ethynylphenylalanine enantiomers »
Z. BENFODDA, D. BENIMELIS, M. JEAN, J.‑V. NAUBRON, V. ROLLAND, P. MEFFRE Amino Acids (2015) 47:899-907 (published online 25 january 2015). DOI 10.1007/s00726-015-1917-1
IF(2014)=3,293

2014

« Synthesis of Cis-5-Trifluoromethylproline from L-Glutamic Acid »
S. ORTIAL, R. DAVE,  Z. BENFODDA, D. BENIMELIS, P. MEFFRE Synlett (2014) 25 : 569-573.
IF (2014)=2,419

2013

« Metabolic intervention on lipid synthesis converging pathways abrogates prostate cancer growth », V. FRITZ, Z. BENFODDA, C. HENRIQUET, S. HURE, J.-P. CRISTOL, F. MICHEL, M.-A. CARBONNEAU, F. CASAS,  L. FAJAS. Oncogene 325101-5110 (2013). IF=6,38.

2012

“Chemoenzymatic routes to enantiomerically pure 2-azatyrosine and 2-, 3- and 4-pyridylalanine derivatives”, A. MOUSSA, P. MEFFRE, J. MARTINEZ,V. ROLLAND. Amino Acids, 42, 1339–1348 (2012) (published online 29 january 2011). DOI 10.1007/s00726-010-0829-3
IF=4,106. 

2011

« Preparation of piperazine derivatives as inhibitors of stearoyl-CoA-desaturase-1 enzyme », L. FAJAS, Z. BENFODDA, V. FRITZ (Brevet, 2011)) , Pub. No:  WO 2011030312 A1 20110317.

“New developements in the synthesis of acetylenic analogues of glutamate”. P. MEFFRE, Z. BENFODDA, D. BENIMELIS, V. ROLLAND, F.C. ACHER. Amino Acids41, supplement 1, S79 (2011) (12th International Congress on Amino Acids, Peptides and Proteins, August 1-5th, 2011, Beijing (PR China), proceeding.
IF=4,106.

2010

“Synthesis and investigation of inhibition effect of fluorinated sulfonamides derivatives on carbonic anhydrase”, Z. BENFODDA, F. GUILLEN, B. ROMESTAND, A. DAHMANI, H. BLANCOU. Eur. J. Med. Chem. 45 1225-1229 5 (2010). IF = 3,269.

 “Abrogation of de novo lipogenesis by Stearoyl Coenzyme A Desaturase 1 inhibition interferes with oncogenic signaling and blocks prostate cancer progression in mice”, Z. BENFODDA*, V. FRITZ*, G. RODIER, C. HENRIQUET, F. IBORRA, C. AVANCES, Y. ALLORY, A. DELATAILLE, S. CULINE, H. BLANCOU, J-P. CRISTOL, F. MICHEL, C. SARDET, L. FAJAS. Mol. Cancer Ther. 9(6) 1740-1754 (2010). (*Z. Benfodda and V. Fritz contributed equally to this work). IF = 4,953.

2009

“A new method for the chlorination of thiocyanates”. Z. BENFODDA, F. GUILLEN, H. ARNION, A. DAHMANI, H. BLANCOU. Heteroatom Chem. 20(6) 355-361 (2009). IF=0.877.

2008

“Synthesis of symmetric and dissymmetric bisperfluoroalkanesulfonylimides. Evaluation of their inhibition on bovine carbonic anhydrase”. Z. BENFODDA, F. GUILLEN, H. BLANCOU. Heteroatom Chem. 19 (5) 542-548 (2008). IF =0.877

2007

“Synthesis of acetylenic analogues of glutamate”. P. MEFFRE, Z. BENFODDA, D. BENIMELIS, F.C. ACHER. Amino acids33, pages LXIV- LXIV (2007). 10th International Congress on Aminoacids, August 20-25th, 2007, Kalithea, Chalkidiki (Greece), proceeding. IF=3,877.

“New synthesis of polyfluoroalkylsulfonylureas”. Z. BENFODDA, L. DELON, F. GUILLEN, H. BLANCOU. J. Fluorine. Chem. 128 (11) 1353-1358 (2007). IF=1,730.

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